Evidence mapPaperPMID 42347882Full record

ArticleClinical cancer research : an official journal of the American Association for Cancer Research2026

A Phase 2 Feasibility Study Combining Pembrolizumab and Metformin in patients with Metastatic Head and Neck Cancer.

Olga Zamulko, Sam Nusbaum, Andrew Osterburg, McKenzie Crist, Maria Lehn, Ilaina Monroe, Audrey Romano, Casey L Allen, Allie Forsythe, Muhammad Kashif Riaz and 7 more

Registry-linked trialAbstract read
In one paragraph

Article in Clinical cancer research : an official journal of the American Association for Cancer Research, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. It is linked to trial NCT04414540 (A Phase 2 Feasibility Study Combining Pembrolizumab and Metformin to Harness the Natural Killer Cytotoxic Response in Metastatic Head and Neck Cancer Patients), which is not on this map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

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The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

NCT04414540 phase2active not recruitingnot on this map

A Phase 2 Feasibility Study Combining Pembrolizumab and Metformin to Harness the Natural Killer Cytotoxic Response in Metastatic Head and Neck Cancer Patients

TypeinterventionalSponsorTrisha Wise-DraperRan2020 to 2026Enrolled21ConditionsHead and Neck Squamous Cell CarcinomaArmsMetformin Extended Release Oral Tablet, Pembrolizumab
3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

17 authors.

Olga ZamulkoUniversity of Cincinnati Cincinnati, Ohio United States.ORCID 0000-0001-5769-7425
Sam NusbaumUniversity of Cincinnati Cincinnati, OH United States.ORCID 0009-0006-1871-8362
Andrew OsterburgUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0003-3018-9134
McKenzie CristUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0001-9271-0322
Maria LehnUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0001-8400-7733
Ilaina MonroeUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0001-8735-7042
Audrey RomanoUniversity of Cincinnati Cincinnati, OH United States.ORCID 0009-0008-2553-681X
Casey L AllenUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0003-3208-5320
Allie ForsytheUniversity of Cincinnati Medical Center Cincinnati, Ohio United States.ORCID 0009-0009-9802-3502
Muhammad Kashif RiazUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0003-1855-7862
Christopher LemmonUniversity of Cincinnati Medical Center Cincinnati, Ohio United States.ORCID 0000-0003-4223-5847
Vinita TakiarUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0002-2499-3516
Jianmin PanUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0002-5998-3481
Shesh N RaiUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0002-8377-353X
Michael BorchersUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0002-8939-3327
Dalia El-GamalUniversity of Cincinnati Medical Center Cincinnati, OH United States.ORCID 0000-0002-1083-8283
Trisha Wise-DraperUniversity of Cincinnati Cincinnati, OH United States.ORCID 0000-0002-7279-4028

Funding

Optimization of peripheral blood mononuclear cell (PBMC) processing for robust downstream functional immune cell analysis and correlation with therapeutic efficacyU01CA267985 · UNIVERSITY OF CINCINNATI · 2025 to 2025
$370k
NCI NIH HHS U01 CA267985
6 · The paper itself

Abstract

backgroundSurvival for recurrent/metastatic head and neck squamous cell carcinoma (R/M HNSCC) remains low with <20% immunotherapy response. Metformin increases tumor-infiltrating CD8+ T and natural killer (NK) cells, which harbor PD-1. In this Phase 2 clinical trial (NCT04414540), we combined metformin and pembrolizumab to evaluate the overall response rate (ORR) in R/M HNSCC and assess NK cell activity.

methodsEligible patients were randomized 1:1 into two arms: (1) metformin ER dose escalation to 2000 mg over 14 days followed by combination with pembrolizumab 200 mg q3 weeks or (2) pembrolizumab 200 mg q3 weeks followed by combination with metformin ER 2000 mg daily. The primary endpoint was ORR per RECIST 1.1. Nineteen evaluable patients were planned to estimate the proportion of approximately 32% ORR. Safety was evaluated by CTCAE v5.0. The distribution, activation, and cytotoxic function of NK cells was analyzed by flow cytometry.

resultsTwenty-one patients were enrolled. 76% were male, 52% smokers, and median age was 64. Ten patients had oropharyngeal tumors, of which 9 were p16 positive. Eighteen patients were evaluable for response, including 4 complete and 5 partial responses for an ORR of 50% (95%CI [29,71]). Combination therapy was well tolerated with no unexpected adverse events (AEs). Five Grade 3 AEs occurred, including nausea, diarrhea, fatigue, and weight loss. Metformin led to increased peripheral NK cell maturation and cytotoxic ability.

conclusionThe combination of metformin and pembrolizumab was well tolerated with mild GI-associated AEs and promising activity warranting further investigation in a randomized trial.

Identifiers

PMID42347882
PMCPMC13436289

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Registered trials

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.