Evidence mapPaperPMID 42426424Full record

ArticleEuropean journal of clinical pharmacology2026

Physiologically based pharmacokinetic modeling of cefotaxime to inform pediatric dosing in renal impairment.

Najia Rahim, Muhammad Sarfraz, Muhammad Wahajuddin

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Article in European journal of clinical pharmacology, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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2 · The registry

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3 · Its place in the literature

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4 · The record

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5 · Who and what money

Authors and funding

3 authors.

Najia RahimDepartment of Pharmacy Practice, Dow College of Pharmacy, Dow University of Health Sciences, Karachi, Sindh, Pakistan. najia.rahim@duhs.edu.pk.ORCID http://orcid.org/0000-0002-9874-8134
Muhammad SarfrazCollege of Pharmacy, Al Ain University, Al Ain, Abu Dhabi, United Arab Emirates.ORCID http://orcid.org/0000-0002-0516-4966
Muhammad WahajuddinInstitute of Cancer Therapeutics, School of Pharmacy & Medical Sciences, Faculty of Life Sciences, University of Bradford, Bradford, West Yorkshire, United Kingdom. m.wahajuddin@bradford.ac.uk.ORCID http://orcid.org/0000-0003-3362-7558

Funding

Scheme for Promotion of Academic and Research Collaboration P3345, P4008 and P 4072
6 · The paper itself

Abstract

backgroundCefotaxime (CFT) is a broad spectrum, third-generation cephalosporin antibiotic prescribed for the treatment of severe infections, yet dosing guidelines for pediatric with renal impairment is scarce. The current study aimed to develop a physiological based pharmacokinetic (PBPK) model to characterize CFT disposition and model-based recommend dose adjustments in pediatrics with renal impairment.

methodsInitially, the PBPK model of CFT was developed in adults with normal renal function before being scaled to pediatrics, considering age-related physiological changes using GastroPlus® software. Renal impairment was modelled through optimization of tubular secretion and glomerular filtration parameters based on observed data for both adults and pediatric populations.

resultsThe model reasonably reproduced the observed pharmacokinetic profiles and showed acceptable agreement with the data (fold error ranges 0.84-1.37) or with renal impairment (fold error ranges 0.87-1.12). When compared to children with normal renal function, the predicted AUC0-∞ in children with renal impairment increased to 1.22- and 1.89-fold for moderate and severe renal impairment, respectively. Model-informed dose recommendations were 60% and 48% of the standard pediatric dose for moderate and severe renal impairment, respectively.

conclusionThis PBPK framework supports rational, model-informed dosing of CFT in pediatric patients with varying renal impairment and supports dose recommendation development for high-risk populations.

Indexed as

Anti-Bacterial AgentsCefotaximeModels, BiologicalRenal InsufficiencyAdolescentAdultArea Under CurveChildChild, PreschoolDose-Response Relationship, DrugFemaleGlomerular Filtration RateHumansInfantMaleThird Generation CephalosporinsAnti-Bacterial AgentsCefotaximeThird Generation CephalosporinsCefotaximeDose recommendationsPBPK modelingRenal impairment

Identifiers

PMID42426424
PMCPMC13350114

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.