Evidence mapPaperPMID 42429358Full record

ArticleThe Journal of organic chemistry2026

Synthesis of Aryl and Heteroaryl Diazophosphonates via Palladium-Catalyzed Cross-Coupling and Their Application in Rhodium-Catalyzed Cyclopropanation.

Yasir Naeem, Duc Ly, Huw M L Davies

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Article in The Journal of organic chemistry, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

3 authors.

Yasir NaeemDepartment of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.ORCID 0000-0003-1448-263X
Duc LyDepartment of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.ORCID 0000-0002-0829-5080
Huw M L DaviesDepartment of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States.ORCID 0000-0001-6254-9398

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Aryl and heteroaryl diazophosphonates are valuable intermediates in organic synthesis and medicinal chemistry. This study presents an efficient and versatile strategy for their synthesis via palladium-catalyzed cross-coupling reactions using readily available diazophosphonate precursors and diverse aryl- and heteroaryl iodides. The method demonstrates excellent yields, broad functional group tolerance, and scalability. Notably, the synthetic utility of the resulting diazophosphonates is showcased through a rhodium-catalyzed cyclopropanation, yielding complex cyclopropane derivatives with high diastereo- and enantioselectivity. Highly enantioselective cyclopropanation was also feasible. This combined palladium- and rhodium-catalyzed approach offers a robust, scalable, and stereoselective pathway for accessing multifunctional scaffolds, thereby expanding the capabilities of modern synthetic chemistry.

Identifiers

PMID42429358
PMCPMC13411051

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.