Evidence map›Paper›PMID 42435652›Full record

ArticleRedox biology2026

Melatonin reprograms antioxidant defenses to suppress ferroptosis via Homer1a/mGluR1-Nrf2/xCT signaling after retinal ischemia-reperfusion.

Ya-Nan Dou, Yuwen Wen, Yuan Huang, Xiuquan Wu, Zehan Zhang, Guanyi Wang, Wangshu Chao, Dongyu Wei, Weihao Lv, Xiaowei Fei and 2 more

Abstract read
In one paragraph

Article in Redox biology, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
–field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

12 authors.

Ya-Nan DouDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Yuwen WenState Key Laboratory of Ophthalmology, Guangdong Provincial Key Laboratory of Ophthalmology and Visual Science, Zhongshan Ophthalmic Center, Sun Yat-sen University, Guangzhou, China.
Yuan HuangDepartment of Ophthalmology, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Xiuquan WuDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Zehan ZhangDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Guanyi WangDepartment of Orthopedic Surgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Wangshu ChaoDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Dongyu WeiCenter of Clinical Aerospace Medicine, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Weihao LvDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China.
Xiaowei FeiDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China. Electronic address: fxwneurosurgery@sina.com.
Zhou FeiDepartment of Neurosurgery, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China. Electronic address: feizhou@fmmu.edu.cn.
Fei FeiDepartment of Ophthalmology, Xijing Hospital, Air Force Military Medical University, Xi'an, Shaanxi, 710032, China. Electronic address: feepluss@fmmu.edu.cn.

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

Melatonin (Mel) exerts antioxidant and anti-ferroptosis effects not only via the canonical receptors Mt1/Mt2 but also via metabotropic glutamate receptor 1 (mGluR1)/glutamate-mediated signaling. Nevertheless, the regulatory mechanism by which Mel modulates mGluR1/glutamate signaling in retinal ischemia-reperfusion (I/R) injury and its downstream effects on ferroptosis and oxidative stress remain poorly understood. Here, bulk RNA sequencing identified that the Mel receptors Mt1/Mt2 and ferroptosis/iron-redox regulators (Gpx4, Fth1, and xCT) were significantly downregulated after retinal I/R. Mel improved retinal structural and visual function, visual-guidance behavior, and electrophysiological responses following I/R while concurrently reducing ferroptotic and inflammatory injury markers. These benefits were largely abolished by Mel membrane receptor antagonists. Mechanistically, Mel upregulated Homer1a in vivo and in vitro in a receptor-dependent manner. Conditional deletion of Homer1a in transgenic mice, as well as Homer1a knockdown in retinal ganglion cells (RGCs), abolished the protective effects of Mel on visual function, along with its anti-ferroptotic and anti-inflammatory activities. Molecular docking and immunoprecipitation assays demonstrated that Mel restored the interaction between Homer1a and mGluR1 and activated the xCT/GSH/Gpx4 antioxidant axis. Pharmacologic inhibition of xCT with the buthionine sulfoximine (BSO) simulation pr genetic interference with xCT expression counteracted the protective effects of Mel. Mel also enhanced Nrf2-mediated transcriptional expression of cCT in a Homer1a/mGluR1-dependent manner. Collectively, our results define a Mel-Homer1a/mGluR1-Nrf2/xCT signaling cascade that promotes RGCs survival after I/R by suppressing ferroptosis/iron-redox reactions, thereby providing a potential translatable strategy for receptor-targeted intervention in I/R-related retinal damage.

Indexed as

AntioxidantsFerroptosisHomer Scaffolding ProteinsMelatoninReceptors, Metabotropic GlutamateReperfusion InjuryRetinal DiseasesAmino Acid Transport System y+AnimalsMiceNF-E2-Related Factor 2Oxidative StressRetinaRetinal Ganglion CellsSignal TransductionAmino Acid Transport System y+AntioxidantsHomer1 protein, mouseHomer Scaffolding ProteinsMelatoninmetabotropic glutamate receptor type 1Nfe2l2 protein, mouseNF-E2-Related Factor 2Receptors, Metabotropic GlutamateSlc7a11 protein, mouseFerroptosisHomer1a/mGluR1Ischemia-reperfusionMelatoninNrf2

Identifiers

PMID42435652
PMCPMC13377451

What Socratic holds

Textmetadata
LicenceCC BY-NC
Read underepoch 390

Registered trials

None linked

Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.