Evidence map›Paper›PMID 42440252›Full record

ArticleDrug delivery and translational research2026

M2 macrophage-derived small extracellular vesicles carrying canagliflozin attenuate experimental asthma.

Yue Zhang, Yile Liu, Lingli Chen, Yating Chen, Xiangrong Zheng

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Article in Drug delivery and translational research, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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4 · The record

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5 · Who and what money

Authors and funding

5 authors.

Yue ZhangDepartment of Pediatrics, Xiangya Hospital, Central South University, Hunan, 410008, China.
Yile LiuDepartment of Pediatrics, Xiangya Hospital, Central South University, Hunan, 410008, China.
Lingli ChenDepartment of Pediatrics, Xiangya Hospital, Central South University, Hunan, 410008, China.
Yating ChenDepartment of Pediatrics, Xiangya Hospital, Central South University, Hunan, 410008, China.
Xiangrong ZhengDepartment of Pediatrics, Xiangya Hospital, Central South University, Hunan, 410008, China. xrzheng@csu.edu.cn.

Funding

the Degree and Postgraduate Education Reform Project of Central South University 2023JGB116the Fundamental Research Funds for the Central Universities of Central South University 2023ZZTS0897the National Natural Science Foundation of China 82170019
6 · The paper itself

Abstract

backgroundAsthma is a chronic inflammatory disorder characterized by immune dysregulation and structural remodeling of the airways, and current therapies remain insufficient, particularly for patients with refractory asthma. Emerging evidence highlights the importance of immunomodulation and local pulmonary administration in improving therapeutic outcomes. Hence, we developed M2 macrophage-derived small extracellular vesicles (M2-sEVs) carrying canagliflozin (CANA) for asthma.

methodsM2-sEVs were isolated and loaded with CANA via ultrasonication to generate CANA-M2-sEVs. The vesicles were characterized by transmission electron microscopy, dynamic light scattering, zeta potential measurement, and sEV-associated marker analysis. Cellular uptake was evaluated using fluorescence imaging. Therapeutic efficacy was assessed in an ovalbumin (OVA)-induced murine asthma model through histological analysis, cytokine profiling, and gene expression assays. The involvement of the PI3K/AKT signaling pathway was investigated using western blotting and pharmacological modulation.

resultsCANA-M2-sEVs retained vesicular morphology and showed nanoscale size distribution with mildly negative surface charge. CANA-M2-sEVs showed efficient, time-dependent cellular uptake in vitro and exerted therapeutic effects following pulmonary administration in vivo. In vivo, CANA-M2-sEVs significantly alleviated airway inflammation, reduced eosinophilic infiltration, and suppressed Th2-associated cytokine production. Moreover, airway remodeling features, including goblet cell metaplasia and collagen deposition, were markedly attenuated. Mechanistically, CANA-M2-sEVs effectively inhibited PI3K and AKT phosphorylation, while pharmacological activation of this pathway partially reversed their anti-inflammatory effects, supporting the involvement of this pathway.

conclusionThis study suggests that CANA-associated M2-sEVs exert anti-inflammatory and anti-remodeling effects in experimental asthma, partly associated with suppression of PI3K/AKT signaling.

Indexed as

AsthmaCanagliflozin (CANA)M2 macrophagesPI3K/AKT signalingSmall extracellular vesicles (sEVs)

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.