Evidence mapPaperPMID 42500704Full record

ArticleSmart molecules : open access2026

Redox-responsive dual-drug nanomedicine integrating cisplatin and trypsin for synergistic reversal of tumor chemoresistance.

Xiaolan Yin, Qi Wang, Ming Zhang, Cheng Zhang, Qixian Chen, Haidong Li, Yan Zhao, Yue Wang, Jingyun Wang, Liuwei Zhang and 1 more

Abstract read
In one paragraph

Article in Smart molecules : open access, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

0numbers the graph read from it
0cells of the map it votes in
0citing papers in PubMed
field-weighted citation impact
1 · What the graph read from it

What it found

Each row is one number read from the abstract, on the scale the paper reported it, with its interval. Left of the dashed line favours the treatment, right favours the comparator. Under each row is the sentence it came from. New to these charts? A ten-minute tutorial.

The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

The trial behind it

Trials whose registry record cites this paper, or whose number appears in the abstract. A trial that started after this paper was published is citing it as background, not reporting it.

Neither the registry nor the abstract names a trial number. If this is a trial report, that itself is worth knowing.

3 · Its place in the literature

Who cites it

0 citing papers in PubMed.

No citing paper in PubMed yet.

4 · The record

Corrections and comments

PubMed lists nothing against this paper. Absence here is not a guarantee, only a check that was made.

5 · Who and what money

Authors and funding

11 authors.

Xiaolan YinSchool of Bioengineering Dalian University of Technology Dalian China.
Qi WangSchool of Bioengineering Dalian University of Technology Dalian China.
Ming ZhangSchool of Bioengineering Dalian University of Technology Dalian China.
Cheng ZhangSchool of Bioengineering Dalian University of Technology Dalian China.
Qixian ChenProvincial Key Laboratory of Interdisciplinary Medical Engineering for Gastrointestinal Carcinoma Liaoning Cancer Hospital & Institute Shenyang China.
Haidong LiSchool of Bioengineering Dalian University of Technology Dalian China.
Yan ZhaoDepartment of Gastric Surgery Cancer Hospital of Dalian University of Technology Shenyang China.
Yue WangDepartment of Gastric Surgery Cancer Hospital of Dalian University of Technology Shenyang China.
Jingyun WangSchool of Bioengineering Dalian University of Technology Dalian China.
Liuwei ZhangInnovation Center of Yangtze River Delta Zhejiang University Jiaxing China.
Hongyan CuiInnovation Center of Yangtze River Delta Zhejiang University Jiaxing China.ORCID https://orcid.org/0000-0002-9386-9287

Funding

No grant is acknowledged in the PubMed record.

6 · The paper itself

Abstract

To overcome cisplatin resistance without increasing systemic toxicity, we rationally elaborated a glutathione-activatable prodrug nanomedicine that chemically co-encapsulates cisplatin and a masked protease. First, a redox-labile succinimide linker (NC-ss-COOH) was covalently grafted onto the ε-amino groups of trypsin to create a "pro-protease" (ssTrypsin) whose catalytic activity is completely silenced in circulation but instantly restored (≥96%) upon cleavage by intratumoral GSH. Simultaneously, cisplatin was stably coordinated to the carboxyl-rich backbone of cRGD-PEG-polyglutamic acid and carboxyl-rich ssTrypsin, forming a polymer-Pt(II) prodrug that prevents premature Pt-GSH adduct formation. These two prodrugs co-self-assemble into potent anti-tumor nanoconstructs that actively target α

Indexed as

cisplatinprotein prodrugreversal of tumor resistancetumor targeting

Identifiers

PMID42500704
PMCPMC13398630

What Socratic holds

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Registered trials

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.