Evidence mapPaperPMID 42589792Full record

ArticlePolymers2026

Development and Optimization of Sodium Deoxycholate-Stabilised Shellac-Based Polymeric Nanoparticles for Enhanced Pharmacokinetics and Anticancer Activity of Etodolac in Hepatocellular Carcinoma.

Ritesh A Fule, Aishwarya S Rangurwar, Pankaj D Nagpure, Helal G Alanazi, Mohammed M Alruwaili, Md Ali Mujtaba, Gamal Osman Elhassan, Siham Abdoun

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Article in Polymers, 2026. The graph could read no effect estimate from its abstract, so it casts no vote on the map. Not yet cited in PubMed.

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1 · What the graph read from it

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The abstract states no effect estimate the extractor could read, or names no intervention and outcome on the map, so this paper lights no cell and moves no belief. It is still indexed, cited and linked below.

2 · The registry

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3 · Its place in the literature

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4 · The record

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5 · Who and what money

Authors and funding

8 authors.

Ritesh A FuleDepartment of Pharmaceutical Science, Dadasaheb Balpande College of Pharmacy, Rashtrasant Tukadoji Maharaj Nagpur University, Nagpur 440037, Maharashtra, India.ORCID 0000-0003-1898-2957
Aishwarya S RangurwarDepartment of Pharmaceutical Science, Dadasaheb Balpande College of Pharmacy, Rashtrasant Tukadoji Maharaj Nagpur University, Nagpur 440037, Maharashtra, India.
Pankaj D NagpureDepartment of Pharmaceutical Science, Dadasaheb Balpande College of Pharmacy, Rashtrasant Tukadoji Maharaj Nagpur University, Nagpur 440037, Maharashtra, India.ORCID 0009-0002-0472-2679
Helal G AlanaziDepartment of Medical Laboratory, College of Applied Medical Sciences, Prince Sattam bin Abdulaziz University, Al-Kharj 11942, Saudi Arabia.ORCID 0009-0004-3843-1137
Mohammed M AlruwailiDepartment of Medical Laboratory Technology, College of Applied Medical Sciences, Northern Border University, Arar 73213, Saudi Arabia.ORCID 0000-0003-2811-4387
Md Ali MujtabaCenter for Health Research, Northern Border University, Arar 73213, Saudi Arabia.ORCID 0000-0002-6372-890X
Gamal Osman ElhassanDepartment of Pharmaceutics, College of Pharmacy, Qassim University, Buraidah 51452, Saudi Arabia.
Siham AbdounDepartment of Pharmaceutics, College of Pharmacy, Qassim University, Buraidah 51452, Saudi Arabia.

Funding

Northern Border University NBU-CRP-2026-2474
6 · The paper itself

Abstract

BACKGROUND/

objectivesHepatocellular carcinoma, or liver cancer, is the sixth most common cancer worldwide and the third leading cause of cancer-related mortality. Therefore, this study aimed to develop and optimise etodolac-loaded sodium deoxycholate-stabilised shellac-based polymeric nanoparticles (ETD-SDS-SHNPs) to improve the pharmacokinetic profile of etodolac (ETD) in HepG2 human hepatocellular carcinoma (HCC) cells.

methodsThe nanoprecipitation method was used to prepare ETD-SDS-SHNPs, which were then optimised using a Box-Behnken design and evaluated for particle size (PS), zeta potential (ZP), entrapment efficiency (EE), solid-state characterization, and in vitro drug dissolution. Furthermore, in vivo oral bioavailability, cytotoxicity, cellular uptake, and cell cycle progression were assessed.

resultsThe optimised ETD-SDS-SHNPs formulation showed an average PS of 192 ± 1.50 nm, ZP of -20.2 ± 0.4 mV, and EE of 81.6 ± 1.42%. Differential scanning calorimetry and X-ray diffraction confirmed the reduced crystallinity of ETD-SDS-SHNPs, indicating partial amorphisation of the drug in the formulation. Field-emission scanning electron microscopy revealed predominantly spherical nanoparticles with relatively smooth surfaces. The peak plasma concentration (C

conclusionsETD-SDS-SHNPs formulation offers an enhanced passive, efficient, and safer nanocarrier platform for repurposing etodolac in liver cancer therapy, showing significant promise for improving clinical outcomes in HCC treatment.

Indexed as

bioavailabilitycytotoxicityetodolachepatocellular carcinomananoparticlesshellac

Identifiers

PMID42589792
PMCPMC13468417

What Socratic holds

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Read under generation 80e0d062 · epoch 390. Bibliography from PubMed, PubMed Central and OpenAlex; grants from NIH RePORTER; trial links from ClinicalTrials.gov; estimates, votes and beliefs from the Socratic graph.